Protein | Organism | No. of ligands tested | No. of good curves | No. of + veashifts/% + veashifts | Best hit (NSC) | ΔTm(°C) | KD(nM)b | Best hit structure |
---|---|---|---|---|---|---|---|---|
DHFR | E. coli | 83 | 32 | 15/46.9 | 309401 | 30.74 | 48.21 |
|
1000006 | H. sapiens | 59 | 43 | 6/13.9 | 133351 | 16.76 | 168.29 |
|
1000001 | R. norvegicus | 86 | 42 | 10/23.8 | 134137 | 12.30 | 406.0 |
|
TrpRS | H. sapiens | 94 | 12 | 5/41.7 | 750690 | 14.57 | 1277.51 |
|
UCE | P. falciparum | 80 | 51 | 2/03.9 | 93427 | 14.86 | 1376.09 |
|
TP2 | P. falciparum | 67 | 12 | 2/16.7 | 106231 | 5.7 | 40872.77 |
|
cDPK | H. sapiens | 80 | 19 | 3/15.8 | 27032 | 2.95 | 48538.90 |
|
NAP 1 | P. knowlesi | 82 | 54 | 4/07.4 | 36398 | 2.21 | 180135.58 |
|