Uniprot ID | Target protein name | Associated bioactivities (Y) | Total number of observations (N-retrieved) | Total number of observations (N-processed) |
---|---|---|---|---|
Q05586 | Glutamate [NMDA] receptor | IC50 | 512 | 320 |
Q99720 | Sigma non-opioid intracellular receptor 1 (Sigma1R) | IC50 | 1895 | 762 |
Q99720 | Sigma non-opioid intracellular receptor 1 (Sigma1R) | Ki | 2584 | 1465 |
CHEMBL613288 (Uniprot ID NA.) | Sigma non-opioid intracellular receptor 2 (Sigma2R) | Ki | 553 | 497 |
P08588 | Beta-1 adrenergic receptor (ADRB1) | IC50 | 1471 | 599 |
P07550 | Beta-2 adrenergic receptor (ADRB2) | IC50 | 1424 | 554 |
P13945 | Beta-3 adrenergic receptor (ADRB3) | EC50 | 1478 | 1227 |
P35348 | Alpha-1A adrenergic receptor | Ki | 1650 | 1260 |
P35368 | Alpha-1b adrenergic receptor | Ki | 1567 | 1260 |
P25100 | Alpha-1D adrenergic receptor | Ki | 2076 | 1060 |
P35367 | Histamine H\(_1\) receptor (HRH1) | Ki | 2239 | 1222 |
P25021 | Histamine H\(_2\) receptor (HRH2) | Ki | 1218 | 385 |
Q9Y5N1 | Histamine H\(_3\) receptor (HRH3) | Ki | 3799 | 3101 |
Q9H3N8 | Histamine H\(_4\) receptor (HRH4) | Ki | 1486 | 1095 |
Q12809 | Potassium voltage-gated channel subfamily H member 2 (HERG) | Ki | 2539 | 1481 |
P21728 | D(1A) dopamine receptor (DRD1) | Ki | 2244 | 1087 |
P14416 | D(2) dopamine receptor (DRD2) | IC50 | 1667 | 725 |
P35462 | D(3) dopamine receptor (DRD3) | IC50 | 1174 | 326 |
P21917 | D(4) dopamine receptor (DRD4) | Ki | 3409 | 1900 |
P21918 | D(1B) dopamine receptor (DRD5) | Ki | 529 | 341 |
P47898 | 5-Hydroxytryptamine receptor 5A | Ki | 382 | 302 |
P50406 | 5-Hydroxytryptamine receptor 6 | Ki | 4084 | 2632 |
P46098 | 5-Hydroxytryptamine receptor 3A | Ki | 517 | 432 |
P28222 | 5-Hydroxytryptamine receptor 1B | Ki | 1129 | 938 |
P41595 | 5-Hydroxytryptamine receptor 2B | Ki | 2034 | 1149 |
P28335 | 5-Hydroxytryptamine receptor 2C | Ki | 3433 | 2157 |
P28221 | 5-Hydroxytryptamine receptor 1D | Ki | 1153 | 973 |
P08908 | 5-Hydroxytryptamine receptor 1A | Ki | 4008 | 3244 |
Q13639 | 5-Hydroxytryptamine receptor 4 | Ki | 540 | 422 |
P34969 | 5-Hydroxytryptamine receptor 7 | Ki | 1753 | 1438 |